Recent developments in the synthesis of hybrid antimalarial drug discoveryArticle Published on 2023-10-312024-09-09 Journal: Bioorg Chem [Category] 말라리아, [키워드] 1,2,3-Triazole 4-Amino-7-chloroquinoline antimalarial Artemisinin Chloroquine Hybrid. PMC 바로가기
In Silico Studies of Four Compounds of Cecropia obtusifolia against Malaria ParasiteArticle Published on 2023-10-032024-08-28 Journal: Molecules [Category] 말라리아, [키워드] antimalarial Cecropia obtusifolia molecular docking molecular dynamics pharmacokinetics Plasmodium
Structure-Activity Relationships and Antiplasmodial Potencies of Novel 3,4-Disubstituted 1,2,5-OxadiazolesArticle Published on 2023-09-232024-08-28 Journal: International Journal of Molecular Sciences [Category] 말라리아, [키워드] 1,2,5-oxadiazoles antimalarial CYP3A4-inhibition Plasmodium falciparum solubility
Influence of amino acid size at the P3 position of N-Cbz-tripeptide Michael acceptors targeting falcipain-2 and rhodesain for the treatment of malaria and human african trypanosomiasisArticle Published on 2023-08-312024-09-10 Journal: Bioorg Chem [Category] 말라리아, [키워드] antimalarial antitrypanosomal Falcipain-2 Michael acceptors neglected tropical diseases Protozoan cysteine proteases Rhodesain. PMC 바로가기
Therapeutical Utilization and Repurposing of Artemisinin and Its Derivatives: A Narrative ReviewArticle Published on 2023-08-312024-09-10 Journal: Adv Biol (Weinh) [Category] 말라리아, [키워드] anticancer antimalarial artemisinin-based drugs coronavirus cytomegalovirus PMC 바로가기
Structural Optimization of BIPPO Analogs as Potent AntimalarialsArticle Published on 2023-06-232024-08-27 Journal: Molecules [Category] 말라리아, [키워드] antimalarial BIPPO analogs structural optimization.
Antioxidant activities of artesunate-procyanidin hybrid compound in erythrocyte and liver of Plasmodium berghei NK65-infected micearticle Published on 2023-04-302024-09-01 Journal: Fundamental & Clinical Pharmacology [Category] 말라리아, [키워드] antimalarial antioxidants artesunate hybrid compound procyanidin [Article Type] article
Identification of 5-(3-(methylsulfonyl)phenyl)-3-(4-(methylsulfonyl)phenyl)-3H-imidazo[4,5-b]pyridine as novel orally bioavailable and metabolically stable antimalarial compound for further explorationarticle Published on 2023-03-312024-09-01 Journal: Chemical Biology & Drug Design [Category] 말라리아, [키워드] ADME-PK antimalarial docking Imidazopyridine PI4 kinase synthesis [Article Type] article
7- N-Substituted-3-oxadiazole Quinolones with Potent Antimalarial Activity Target the Cytochrome bc1 ComplexArticle Published on 2023-03-102024-08-28 Journal: ACS Infectious Diseases [Category] 말라리아, [키워드] antimalarial cytochrome bc1 malaria Mitochondria Plasmodium
A comprehensive overview of Artemisinin and its derivatives as anticancer agentsarticle Published on 2023-02-282024-09-01 Journal: European Journal of Medicinal Chemistry [Category] 말라리아, [키워드] anticancer antimalarial Artemisinin derivatives mechanism [Article Type] article