Exploring the antimalarial and antioxidant efficacy of transition metal(II) chelates of thiosemicarbazone ligands: spectral investigations, molecular docking, DFT, MESP and ADMETarticle Published on 2024-02-282024-09-01 Journal: BioMetals [Category] 말라리아, [키워드] Antimalarial activity antioxidant activity DFT MESP Spectral technique Thiosemicarbazone ligand [Article Type] article
An Overview on Antimalarial Peptides: Natural Sources, Synthetic Methodology and Biological PropertiesArticle Published on 2023-11-252024-08-29 Journal: Molecules [Category] 말라리아, [키워드] Antimalarial activity Isolation peptide synthesis peptide.
Novel hydrazone derivatives of N-amino-11-azaartemisinin with high order of antimalarial activity against multidrug-resistant Plasmodium yoelii nigeriensis in Swiss mice via intramuscular routearticle Published on 2022-02-282024-09-01 Journal: Bioorganic & Medicinal Chemistry Letters [Category] 말라리아, [키워드] 11-azaartemisnin Antimalarial activity Artemisinin multidrug-resistant [Article Type] article
1,2,3-Triazole derivatives: synthesis, docking, cytotoxicity analysis and in vivo antimalarial activityarticle Published on 2021-12-312024-09-01 Journal: Journal of Biomolecular Nmr [Category] 말라리아, [키워드] 1,2,3-Triazoles compounds Antimalarial activity Cytotoxicity evaluation molecular docking Plasmodium berghei [Article Type] article
Sinigrin in combination with artesunate provides protection against lethal murine malaria via falcipain-3 inhibition and immune modulationarticle Published on 2021-12-312024-09-01 Journal: International Immunopharmacology [Category] 말라리아, [키워드] Antimalarial activity Glucosinolates Plasmodium Sinigrin Thlaspi arvense [Article Type] article
Novel naphthyl based 1,2,4-trioxanes: Synthesis and in vivo efficacy in the Plasmodium yoelii nigeriensis in Swiss micearticle Published on 2021-11-302024-09-01 Journal: Bioorganic & Medicinal Chemistry Letters [Category] 말라리아, [키워드] 1,2,4-trioxane Antimalarial activity endoperoxide multidrug-resistant Photooxygenation β-Hydroxyhydroperoxide [Article Type] article
Synthesis of novel 1,2,4-trioxanes and antimalarial evaluation against multidrug-resistant Plasmodium yoelii nigeriensisarticle Published on 2021-10-312024-09-01 Journal: Bioorganic & Medicinal Chemistry Letters [Category] 말라리아, [키워드] 1,2,4-trioxane Antimalarial activity multidrug-resistant Photooxygenation β-Hydroxyhydroperoxide [Article Type] article
Antiplasmodial, antimalarial activities and toxicity of African medicinal plants: a systematic review of literature아프리카 약용 식물의 항말라리아, 항플라스모디움 활성 및 독성: 문헌에 대한 체계적 검토Research Published on 2021-08-252024-08-08 Journal: Malaria Journal [Category] 말라리아, [키워드] Antimalarial activity Antiplasmodial activity malaria medicinal plants [DOI] 10.1186/s12936-021-03866-0 PMC 바로가기 [Article Type] Research
5-Phenoxy Primaquine Analogs and the Tetraoxane Hybrid as Antimalarial Agents5-페노옥시 프리마퀸 유사체와 테트라옥산 하이브리드 항말라리아제Article Published on 2021-06-302024-08-08 Journal: Molecules [Category] 말라리아, [키워드] Antimalarial activity heme polymerization inhibition activity hybrid drug primaquine structure–activity relationship tetraoxane [DOI] 10.3390/molecules26133991 PMC 바로가기 [Article Type] Article
In silico study, synthesis, and evaluation of the antimalarial activity of hybrid dimethoxy pyrazole 1,3,5-triazine derivativesarticle Published on 2021-03-312024-09-01 Journal: Journal of Biochemical and Molecular Toxicology [Category] 말라리아, [키워드] 1,3,5-triazine Antimalarial activity docking pyrazole synthesis [Article Type] article