Acyloxymethyl and alkoxycarbonyloxymethyl prodrugs of a fosmidomycin surrogate as antimalarial and antibacterial agentsArticle Published on 2023-01-052024-08-29 Journal: European Journal of Medicinal Chemistry [Category] 말라리아, [키워드] ESKAPE fosmidomycin Isoprenoid biosynthesis malaria prodrugs Tuberculosis
Metabolic Survival Adaptations of Plasmodium falciparum Exposed to Sublethal Doses of FosmidomycinArticle Published on 2021-03-182024-08-28 Journal: Med Instrum [Category] 말라리아, [키워드] Apicoplast fosmidomycin genome-scale metabolic model Metabolic modeling metabolomics Plasmodium falciparum prenylation transcriptomics
Predicting Drug Resistance Using Deep Mutational Scanning약물 저항성 예측을 위한 심층 변이 스캐닝Communication Published on 2020-05-112024-08-11 Journal: Molecules [Category] 말라리아, [키워드] drug resistance DXR fosmidomycin Genome editing sequence to activity mapping [DOI] 10.3390/molecules25092265 PMC 바로가기 [Article Type] Communication
Deciphering structure, function and mechanism of Plasmodium IspD homologs from their evolutionary imprintsarticle Published on 2019-04-302024-09-01 Journal: Journal of Computer-Aided Molecular Design [Category] 말라리아, [키워드] Apicoplast drug target Evolutionary imprints fosmidomycin IspD Non-mevalonate pathway Structure–function relationships [Article Type] article
Alternatives to currently used antimalarial drugs: in search of a magic bullet현재 사용되는 항말라리아 약물의 대안: 마법의 총알을 찾아서Article Published on 2016-11-042024-08-12 Journal: Infectious Diseases of Poverty [Category] 말라리아, [키워드] artemisinin derivatives Chemotherapy Drug development fosmidomycin malaria Medicine for malaria venture Novel antimalarial drugs tafenoquine [DOI] 10.1186/s40249-016-0196-8 PMC 바로가기
Whole-Genome Sequencing to Evaluate the Resistance Landscape Following Antimalarial Treatment Failure With Fosmidomycin-ClindamycinArticle Published on 2016-10-012024-08-27 Journal: Nanoscale [Category] 말라리아, [키워드] Clindamycin fosmidomycin malaria Plasmodium recrudescence whole genome amplification.
Fosmidomycin as an antimalarial drug: a meta-analysis of clinical trialsArticle Published on 2015-12-312024-09-10 Journal: Future Microbiol [Category] 말라리아, [키워드] antimalarial drug Clinical studies DOXP reducto-isomerase Drug development fosmidomycin fosmidomycin-clindamycin malaria PMC 바로가기