Ginkgolic acids inhibit SARS-CoV-2 and its variants by blocking the spike protein/ACE2 interplayArticle Published on 2023-01-312023-07-11 Journal: International journal of biological macromolecules [Category] COVID19(2023년), [키워드] ginkgolic acid S-RBD SARS-CoV-2. [DOI] 10.1016/j.ijbiomac.2022.12.057 PMC 바로가기
[Discovery of SARS-CoV-2 main protease inhibitors using an optimized FRET-based high-throughput screening assay]Article Published on 2022-06-252023-07-09 Journal: Sheng wu gong cheng xue bao = Chinese journal of biotechnology [Category] COVID19(2023년), [키워드] fluorescence resonance energy transfer (FRET) ginkgolic acid High-throughput screening Main protease inhibitor plumbagin. SARS-CoV-2 [DOI] 10.13345/j.cjb.210657 PMC 바로가기
Ginkgolic Acid Inhibits Coronavirus Strain 229E Infection of Human Epithelial Lung CellsCommunication Published on 2021-09-262022-10-28 Journal: Pharmaceuticals [Category] COVID-19, [키워드] 229E acid added affected Antiviral antiviral activity Antiviral compound caused coronavirus Coronaviruses COVID-19 pandemic CPE Cytopathic effect deaths demonstrated disrupting Ebola effective effective antiviral treatment Efficacy epithelial Epstein Barr virus exhibited expression fusion inhibitor ginkgolic acid globe HCoV-229E Herpe HIV HSV-1 Human Human coronavirus in vitro in vivo individual Infection influenza A inhibit inhibited inhibiting lung cell Post-infection progeny Proteins reduced reported SARS-CoV-2 significantly similarity strain Vaccine Viral mutations Viral protein Viral proteins virus production viruses [DOI] 10.3390/ph14100980 PMC 바로가기 [Article Type] Communication
Ginkgolic acid and anacardic acid are specific covalent inhibitors of SARS-CoV-2 cysteine proteasesResearch Published on 2021-02-282022-11-01 Journal: Cell & Bioscience [Category] COVID-19, [키워드] 3CL pro addition Anacardic acid antivirals characterized Compound compounds concentrations cysteine protease demonstrated develop enzyme ginkgolic acid in vitro inhibit SARS-CoV-2 inhibitor inhibitors of SARS-CoV-2 mechanism of action natural product nontoxic Papain-like protease Papain‐like protease protease provide Replication Result SARS-CoV-2 the SARS-CoV-2 [DOI] 10.1186/s13578-021-00564-x PMC 바로가기 [Article Type] Research