Synthesis of a Hexavalent Betulinic Acid Derivative as a Hemagglutinin-Targeted Influenza Virus Entry InhibitorArticle Published on 2020-07-062023-06-23 Journal: Molecular Pharmaceutics [Category] 신종인플루엔자, [키워드] betulinic acid Entry inhibitor Influenza virus α-cyclodextrin. [DOI] 10.1021/acs.molpharmaceut.0c00244
Broad-Spectrum Coronavirus Fusion Inhibitors to Combat COVID-19 and Other Emerging Coronavirus DiseasesReview Published on 2020-05-282022-10-29 Journal: International Journal of Molecular Sciences [Category] COVID-19, MERS, SARS, [키워드] acute respiratory syndrome antibodies antibody antiviral drug approved caused characterized combat conserved coronavirus coronavirus disease COVID-19 Disadvantages Diseases drug drugs targeting Entry inhibitor fusion fusion inhibitor inhibitors MERS Middle East Novel coronavirus Other pathogen peptide Protease inhibitor protease inhibitors SARS Coronavirus SARS-CoV-2 syndrome Transmissibility Vaccine Vaccines [DOI] 10.3390/ijms21113843 PMC 바로가기 [Article Type] Review
Characterization of the receptor-binding domain (RBD) of 2019 novel coronavirus: implication for development of RBD protein as a viral attachment inhibitor and vaccine2019 신종 코로나바이러스 수용체 결합 도메인(RBD) 특성 규명: 바이러스 부착 억제제 및 백신으로서의 RBD 단백질 개발에 대한 시사점Article Published on 2020-03-192022-09-06 Journal: Cellular and Molecular Immunology [Category] Communicable Disease, COVID-19, MERS, SARS, [키워드] 2019 novel coronavirus 2019-nCoV ACE2 ACE2 receptor ACE2-expressing cells acute respiratory syndrome acute respiratory syndrome coronavirus acute respiratory syndrome coronavirus 2 angiotensin angiotensin-converting enzyme 2 antibodies binding binding affinity causative agent characterization coronavirus coronavirus disease Coronavirus disease 2019 CoV CoV infection COVID-19 cross-neutralization cross-neutralize SARS-CoV-2 cross-react develop effective Entry inhibitor entry inhibitors enzyme exhibited fusion global public health host cells Human Immunotherapy in viral Infection inhibiting Novel coronavirus outbreak Protein RBD RBD protein Receptor-binding domain receptors respiratory S protein Safe SARS-CoV infection SARS-CoV RBD SARS-CoV RBD-based vaccine SARS-CoV RBD-based vaccines SARS-CoV RBD-induced antisera SARS-CoV RBD-specific antibodies SARS-CoV RBD-specific antibody SARS-CoV-2 SARS-CoV-2 and SARS-CoV infection SARS-CoV-2 RBD SARS-CoV-2 RBD protein SARS-CoV-2 S protein severe acute respiratory syndrome Coronavirus significantly higher specific antibodies Spike protein target the RBD protein the receptor-binding domain Therapeutics Vaccine Vaccines Viral viral attachment inhibitor viral infection viral inhibitor [DOI] 10.1038/s41423-020-0400-4 PMC 바로가기 [Article Type] Article
Development of a mass spectrometric screening assay for hepatitis B virus entry inhibitorsArticle Published on 2020-01-302023-06-09 Journal: Journal of pharmaceutical and biomedical analysis [Category] B형 간염, [키워드] Drug screening Entry inhibitor Hepatitis B virus liquid chromatography-mass spectrometry sodium taurocholate cotransporting polypeptide Taurocholic acid. [DOI] 10.1016/j.jpba.2019.112959
Design, synthesis and biological evaluation of amino acids-oleanolic acid conjugates as influenza virus inhibitorsArticle Published on 2019-12-012023-06-23 Journal: Bioorganic & Medicinal Chemistry [Category] 신종인플루엔자, [키워드] amino acids Entry inhibitor hemagglutinin influenza A virus Oleanolic acid. [DOI] 10.1016/j.bmc.2019.115147
Treatment of chronic hepatitis due to hepatitis B and hepatitis delta virus coinfectionReview Published on 2019-12-012023-06-16 Journal: International journal of antimicrobial agents [Category] B형 간염, [키워드] Entry inhibitor HBsAg release blocker Hepatitis Delta virus IFN-lambda peg-IFN Prenylation inhibitor. [DOI] 10.1016/j.ijantimicag.2019.09.012 [Article Type] Review
Excellent safety and effectiveness of high-dose myrcludex-B monotherapy administered for 48 weeks in HDV-related compensated cirrhosis: A case report of 3 patientsCase Reports Published on 2019-10-012023-06-19 Journal: Journal of hepatology [Category] B형 간염, [키워드] Bulevirtide Coinfection Entry inhibitor HBV HDV HDV RNA Hepatitis Delta Myrcludex-B NTCP T cell [DOI] 10.1016/j.jhep.2019.07.003 [Article Type] Case Reports
Drugs in the Pipeline for HBVReview Published on 2019-08-012023-06-17 Journal: Clinics in Liver Disease [Category] B형 간염, [키워드] cccDNA Core protein inhibitor Entry inhibitor HBV cure Immunotherapy siRNA TLR agonist [DOI] 10.1016/j.cld.2019.04.006 [Article Type] Review
Synthesis, structure activity relationship and in vitro anti-influenza virus activity of novel polyphenol-pentacyclic triterpene conjugatesArticle Published on 2019-02-012023-06-24 Journal: European journal of medicinal chemistry [Category] 신종인플루엔자, [키워드] Entry inhibitor hemagglutinin Influenza virus pentacyclic triterpene polyphenol [DOI] 10.1016/j.ejmech.2018.12.006
Identification of pyrrolo[3,2-c]pyridin-4-amine compounds as a new class of entry inhibitors against influenza viruses in vitroArticle Published on 2016-09-302023-06-21 Journal: Biochemical and Biophysical Research Communication [Category] 조류인플루엔자, [키워드] antiviral drugs Entry inhibitor High-throughput screening Influenza virus Pyrrolopyridinamine. [DOI] 10.1016/j.bbrc.2016.08.162