Azvudine (FNC): a promising clinical candidate for COVID-19 treatmentResearch Highlight Published on 2020-10-102022-10-04 Journal: Signal Transduction and Targeted Therapy [Category] MERS, SARS, 신약개발, 임상, 치료제, [키워드] Azvudine COVID-19 Infectious diseases Target identification Treatment [DOI] 10.1038/s41392-020-00351-z PMC 바로가기 [Article Type] Research Highlight
Salvianolic acid C potently inhibits SARS-CoV-2 infection by blocking the formation of six-helix bundle core of spike proteinLetter Published on 2020-10-062022-10-29 Journal: Signal Transduction and Targeted Therapy [Category] COVID-19, MERS, SARS, [키워드] Drug screening inhibit SARS-COV-2 infection Spike protein Target identification [DOI] 10.1038/s41392-020-00325-1 PMC 바로가기 [Article Type] Letter
Feline coronavirus drug inhibits the main protease of SARS-CoV-2 and blocks virus replicationArticle Published on 2020-08-272022-10-04 Journal: Nature Communications [Category] 변종, 치료제, [키워드] 3CL pro block Cell culture cleavage coronavirus Coronavirus infection COVID-19 crystal structure Cys145 drug candidate drug target effective inhibitor Feline infectious peritonitis inhibit inhibitor inhibitors of SARS-CoV-2 M pro Modification NMR analysis nucleophilic polyprotein proceed protease Protease inhibitor Proteases Replication reveal SARS-CoV SARS-CoV-2 SARS-CoV-2 replication Target identification treat treated Treatment Trial virus virus replication X-ray crystallography [DOI] 10.1038/s41467-020-18096-2 PMC 바로가기 [Article Type] Article
Exploring the SARS-CoV-2 virus-host-drug interactome for drug repurposingArticle Published on 2020-07-142022-10-04 Journal: Nature Communications [Category] SARS, 신약개발, 치료제, [키워드] Algorithm Algorithms candidate Candidates caused coronavirus disease-2019 COVID-19 develop Drivers drug candidates Drug-target interactions Host hypothese Infectious disease information interactions molecular mechanism Network topology pathogenicity platform protein interactions Research resource SARS-CoV-2 SARS-COV-2 infection Scientific community Software Spread Systems biology Target identification the SARS-CoV-2 the SARS-CoV-2 virus time-consuming viral infection Virus life cycle [DOI] 10.1038/s41467-020-17189-2 PMC 바로가기 [Article Type] Article
Numerical evaluation of spray position for improved nasal drug deliveryArticle Published on 2020-06-292022-10-29 Journal: Scientific Reports [Category] Coronavirus, SARS, [키워드] Analysis average Coronavirus infection COVID-19 pandemic disease dose drug drug delivery ENhance healthcare humans in vitro initial knowledge lack Mathematics and computing mitigate mucosa nasal prevalent protocol Respiratory tract diseases significantly Standard-of-care Target identification therapeutic option topical translate Transport Vaccine while [DOI] 10.1038/s41598-020-66716-0 PMC 바로가기 [Article Type] Article
Combining Stage Specificity and Metabolomic Profiling to Advance Antimalarial Drug Discovery단계 특이성과 대사체 프로파일링을 결합하여 항말라리아 약물 발견을 발전시키다Article Published on 2020-02-202024-08-26 Journal: Cell Chemical Biology [Category] 말라리아, [키워드] Asexual blood stages drug resistance hemoglobin catabolism malaria metabolomics Mitochondria mode of action Plasmodium falciparum Target identification [DOI] 10.1016/j.chembiol.2019.11.009 PMC 바로가기 [Article Type] Article
Fusion mechanism of 2019-nCoV and fusion inhibitors targeting HR1 domain in spike proteinCorrespondence Published on 2020-02-112022-11-01 Journal: Cellular and Molecular Immunology [Category] COVID-19, SARS, [키워드] 2019-nCoV fusion HR1 domain inhibitor mechanism Mechanisms of disease Spike protein Target identification [DOI] 10.1038/s41423-020-0374-2 PMC 바로가기 [Article Type] Correspondence
Unpacking ‘Artemisinin Resistance’article Published on 2017-06-302024-09-01 Journal: Trends in Pharmacological Sciences [Category] 말라리아, [키워드] Artemisinin resistance artemisinin targets mechanism of action Target identification [Article Type] article