Synthesis and Biological Evaluation of Honokiol Derivatives Bearing 3-((5-phenyl-1,3,4-oxadiazol-2-yl)methyl)oxazol-2(3H)-ones as Potential Viral Entry Inhibitors against SARS-CoV-2Communication Published on 2021-08-312022-10-28 Journal: Pharmaceuticals [Category] COVID-19, [키워드] 2019 coronavirus disease ACE2 ACE2 blocker activities analogue Antiviral antiviral activity antiviral efficacy antiviral molecules Bearing bind binding binding affinity Biological Biosafety Level 3 BLI caused contribute cortex COVID-19 demonstrated derivative develop effective ELISA assay examined Health Honokiol honokiol analogues host cell human Ace2 protein inhibitor inhibitory effect lower binding energy medication molecular docking parental Potential Research SARS-CoV-2 SARS-CoV-2 pseudovirus SARS-CoV-2 spike SARS-CoV-2 viral SARS-CoV-2 virus infection strain synthesis the SARS-CoV-2 virus Viral entry inhibitors [DOI] 10.3390/ph14090885 PMC 바로가기 [Article Type] Communication
Keep out! SARS-CoV-2 entry inhibitors: their role and utility as COVID-19 therapeutics입장 금지!SARS-COV-2 진입 억제제 : COVID-19 Therapeutics로서의 역할과 유용성Review Published on 2021-07-232022-09-01 Journal: Virology Journal [Category] SARS, 변종, 유전자 메커니즘, 진단, [키워드] antibodies antigenic antigenic drift approval best COVID-19 COVID-19 pandemic COVID-19 therapeutics effective effective vaccine Emerging sarbecoviruses globe Health healthcare herd immunity highlight Immunity individual inhibitor Keep less life management mechanism of action Mild miniprotein Mortality Mutation Neutralizing antibodies neutralizing antibody new SARS-CoV-2 pandemic Population Prophylaxis recombinant ACE2 Sarbecoviruses SARS-CoV-2 SARS-CoV-2 entry SARS-CoV-2 variants significantly the vaccine Therapeutic strategies therapeutic strategy utility vaccinate Vaccine Vaccines variant Viral viral entry Viral entry inhibitors zoonotic sarbecoviruses [DOI] 10.1186/s12985-021-01624-x PMC 바로가기 [Article Type] Review
Plants and Natural Products with Activity against Various Types of Coronaviruses: A Review with Focus on SARS-CoV-2Review Published on 2021-07-052022-10-30 Journal: Molecules [Category] COVID-19, SARS, [키워드] activity angiotensin-converting enzyme inhibitors (ACEi) Antiviral biomolecules caused Coronavirus disease of 2019 (COVID-19) Coronaviruses COVID-19 Evidence focus hospital resources Host human cells individuals management medicinal plants Medicine Middle East respiratory syndrome (MERS) mitigate natural pandemic disease Particular plant plants product RAAS renin–angiotensin–aldosterone system (RAAS) review SARS-CoV-2 severe acute respiratory syndrome coronavirus (SARS-CoV) Symptom System the SARS-CoV-2 the SARS-CoV-2 virus Type various coronaviruses Viral entry inhibitors [DOI] 10.3390/molecules26134099 PMC 바로가기 [Article Type] Review
Bulevirtide for HBV and HDV infectionsArticle Published on 2021-07-012023-06-11 Journal: Drugs of today (Barcelona, Spain : 1998) [Category] B형 간염, [키워드] Bulevirtide HBV/HDV infections hepatitis B Hepatitis D Sodium-bile acid cotransporter inhibitors Viral entry inhibitors Viral hepatitis. [DOI] 10.1358/dot.2021.57.7.3283861 PMC 바로가기